JOSÉ ANTONIO
ESCARIO GARCÍA-TREVIJANO
Profesor emérito
Publicacións nas que colabora con JOSÉ ANTONIO ESCARIO GARCÍA-TREVIJANO (33)
2021
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Promising hit compounds against resistant trichomoniasis: Synthesis and antiparasitic activity of 3-(ω-aminoalkoxy)-1-benzyl-5-nitroindazoles
Bioorganic and Medicinal Chemistry Letters, Vol. 37
2018
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Antichagasic, Leishmanicidal, and Trichomonacidal Activity of 2-Benzyl-5-nitroindazole-Derived Amines
ChemMedChem, Vol. 13, Núm. 12, pp. 1246-1259
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Drug repositioning for novel antitrichomonas from known antiprotozoan drugs using hierarchical screening
Future Medicinal Chemistry, Vol. 10, Núm. 8, pp. 863-878
2016
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Antichagasic and trichomonacidal activity of 1-substituted 2-benzyl-5-nitroindazolin-3-ones and 3-alkoxy-2-benzyl-5-nitro-2H-indazoles
European Journal of Medicinal Chemistry, Vol. 115, pp. 295-310
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In vitro trichomonacidal activity and preliminary in silico chemometric studies of 5-nitroindazolin-3-one and 3-alkoxy-5-nitroindazole derivatives
Parasitology, Vol. 143, Núm. 1, pp. 34-40
2015
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Sequestration of host-CD59 as potential immune evasion strategy of Trichomonas vaginalis
Acta Tropica, Vol. 149, pp. 1-7
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Synthesis and in vitro and in vivo biological evaluation of substituted nitroquinoxalin-2-ones and 2,3-diones as novel trichomonacidal agents
European Journal of Medicinal Chemistry, Vol. 94, pp. 276-283
2014
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A sequential procedure for rapid and accurate identification of putative trichomonacidal agents
Journal of Microbiological Methods, Vol. 105, pp. 162-167
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Antiprotozoan lead discovery by aligning dry and wet screening: Prediction, synthesis, and biological assay of novel quinoxalinones
Bioorganic and Medicinal Chemistry, Vol. 22, Núm. 5, pp. 1568-1585
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Determination of internal transcribed spacer regions (ITS) in Trichomonas vaginalis isolates and differentiation among Trichomonas species
Parasitology International, Vol. 63, Núm. 2, pp. 427-431
2012
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Validation of a modified fluorimetric assay for the screening of trichomonacidal drugs
Memorias do Instituto Oswaldo Cruz, Vol. 107, Núm. 5, pp. 637-643
2009
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Discovery of novel trichomonacidals using LDA-driven QSAR models and bond-based bilinear indices as molecular descriptors
QSAR and Combinatorial Science, Vol. 28, Núm. 1, pp. 9-26
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Synthesis and evaluation of 1,1′-hydrocarbylenebis(indazol-3-ols) as potential antimalarial drugs
ChemMedChem, Vol. 4, Núm. 1, pp. 78-87
2008
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Bond-based linear indices in QSAR: Computational discovery of novel anti-trichomonal compounds
Journal of Computer-Aided Molecular Design, Vol. 22, Núm. 8, pp. 523-540
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New antitrichomonal drug-like chemicals selected by bond (edge)-based TOMOCOMD-CARDD descriptors
Journal of Biomolecular Screening, Vol. 13, Núm. 8, pp. 785-794
2006
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Antiparasitic properties of homoallylamines and related compounds
Acta Parasitologica, Vol. 51, Núm. 1, pp. 73-78
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New ligand-based approach for the discovery of antitrypanosomal compounds
Bioorganic and Medicinal Chemistry Letters, Vol. 16, Núm. 7, pp. 1898-1904
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Predicting antitrichomonal activity: A computational screening using atom-based bilinear indices and experimental proofs
Bioorganic and Medicinal Chemistry, Vol. 14, Núm. 19, pp. 6502-6524
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Selective activity of polyene macrolides produced by genetically modified Streptomyces on Trypanosoma cruzi
International Journal of Antimicrobial Agents, Vol. 28, Núm. 2, pp. 104-109
2005
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A computer-based approach to the rational discovery of new trichomonacidal drugs by atom-type linear indices
Current Drug Discovery Technologies, Vol. 2, Núm. 4, pp. 245-265