BELLINDA
BENHAMÚ SALAMA
Profesora titular de universidad
MARÍA DEL HENAR
VÁZQUEZ VILLA
Profesora contratada doctora
Publicaciones en las que colabora con MARÍA DEL HENAR VÁZQUEZ VILLA (14)
2023
2022
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2-(Fluoromethoxy)-4′-(S-methanesulfonimidoyl)-1,1′-biphenyl (UCM-1306), an Orally Bioavailable Positive Allosteric Modulator of the Human Dopamine D1Receptor for Parkinson's Disease
Journal of Medicinal Chemistry, Vol. 65, Núm. 18, pp. 12256-12272
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Discovery of V-0219: A Small-Molecule Positive Allosteric Modulator of the Glucagon-Like Peptide-1 Receptor toward Oral Treatment for "diabesity"
Journal of Medicinal Chemistry, Vol. 65, Núm. 7, pp. 5449-5461
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New Trends in Aging Drug Discovery
Biomedicines, Vol. 10, Núm. 8
2019
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Allosteric modulators targeting GPCRs
GPCRs: Structure, Function, and Drug Discovery (Elsevier), pp. 195-241
2017
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A Positive Allosteric Modulator of the Serotonin 5-HT2C Receptor for Obesity
Journal of Medicinal Chemistry, Vol. 60, Núm. 23, pp. 9575-9584
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A new serotonin 5-HT 6 receptor antagonist with procognitive activity - Importance of a halogen bond interaction to stabilize the binding
Scientific Reports, Vol. 7
2016
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Chemoproteomic approach to explore the target profile of GPCR ligands: Application to 5-HT1A and 5-HT6 receptors
Chemistry - A European Journal, Vol. 22, Núm. 4, pp. 1313-1321
2014
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Serotonin 5-HT6receptor antagonists for the treatment of cognitive deficiency in Alzheimer's disease
Journal of Medicinal Chemistry, Vol. 57, Núm. 17, pp. 7160-7181
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The extracellular entrance provides selectivity to serotonin 5-HT 7 receptor antagonists with antidepressant-like behavior in vivo
Journal of Medicinal Chemistry, Vol. 57, Núm. 15, pp. 6879-6884
2013
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New serotonin 5-HT1A receptor agonists endowed with antinociceptive activity in vivo
Journal of Medicinal Chemistry, Vol. 56, Núm. 20, pp. 7851-7861
2011
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New serotonin 5-HT 1A receptor agonists with neuroprotective effect against ischemic cell damage
Journal of Medicinal Chemistry, Vol. 54, Núm. 23, pp. 7986-7999
2010
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Development of fluorescent ligands for the human 5-HT1A receptor
ACS Medicinal Chemistry Letters, Vol. 1, Núm. 6, pp. 249-253
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Development of molecular probes for the human 5-HT6 receptor
Journal of Medicinal Chemistry, Vol. 53, Núm. 19, pp. 7095-7106