![Foto de JOSÉ ANTONIO](/img/nophoto.png)
JOSÉ ANTONIO
ESCARIO GARCÍA-TREVIJANO
Profesor emérito
Publicaciones (81) Publicaciones de JOSÉ ANTONIO ESCARIO GARCÍA-TREVIJANO
2024
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Impact of COVID-19 Pandemic on the Trends of Trichomonas vaginalis Infection in a Tertiary Hospital of Madrid, Spain
Microorganisms, Vol. 12, Núm. 3
2022
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5-Nitroindazole-based compounds: further studies for activity optimization as anti-Trypanosoma cruzi agents
Acta Tropica, Vol. 234
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La anfotericina B normalmente es subdosificada en el tratamiento de la leishmaniasis cutánea experimental
Ars pharmaceutica, Vol. 63, Núm. 3, pp. 253-262
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Thio- and selenosemicarbazones as antiprotozoal agents against Trypanosoma cruzi and Trichomonas vaginalis
Journal of enzyme inhibition and medicinal chemistry, Vol. 37, Núm. 1, pp. 781-791
2021
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Promising hit compounds against resistant trichomoniasis: Synthesis and antiparasitic activity of 3-(ω-aminoalkoxy)-1-benzyl-5-nitroindazoles
Bioorganic and Medicinal Chemistry Letters, Vol. 37
2020
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Activity profile of two 5-nitroindazole derivatives over the moderately drug-resistant Trypanosoma cruzi y strain (DTU TcII): In vitro and in vivo studies
Parasitology, Vol. 147, Núm. 11, pp. 1216-1228
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Trichomoniasis in a tertiary hospital of Madrid, Spain (2013–2017): prevalence and pregnancy rate, coinfections, metronidazole resistance, and endosymbiosis
Parasitology Research, Vol. 119, Núm. 6, pp. 1915-1923
2018
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Antichagasic, Leishmanicidal, and Trichomonacidal Activity of 2-Benzyl-5-nitroindazole-Derived Amines
ChemMedChem, Vol. 13, Núm. 12, pp. 1246-1259
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Drug repositioning for novel antitrichomonas from known antiprotozoan drugs using hierarchical screening
Future Medicinal Chemistry, Vol. 10, Núm. 8, pp. 863-878
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Experimental models in Chagas disease: a review of the methodologies applied for screening compounds against Trypanosoma cruzi
Parasitology Research, Vol. 117, Núm. 11, pp. 3367-3380
2017
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Novel Imidazo[4,5-c][1,2,6]thiadiazine 2,2-dioxides as antiproliferative trypanosoma cruzi drugs: Computational screening from neural network, synthesis and in vivo biological properties
European Journal of Medicinal Chemistry, Vol. 136, pp. 223-234
2016
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Antichagasic and trichomonacidal activity of 1-substituted 2-benzyl-5-nitroindazolin-3-ones and 3-alkoxy-2-benzyl-5-nitro-2H-indazoles
European Journal of Medicinal Chemistry, Vol. 115, pp. 295-310
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Biological approaches to characterize the mode of action of two 5-nitroindazolinone prototypes on Trypanosoma cruzi bloodstream trypomastigotes
Parasitology, Vol. 143, Núm. 11, pp. 1469-1478
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In vitro trichomonacidal activity and preliminary in silico chemometric studies of 5-nitroindazolin-3-one and 3-alkoxy-5-nitroindazole derivatives
Parasitology, Vol. 143, Núm. 1, pp. 34-40
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Nuevos métodos "in sílico" y clásicos de selección de moléculas farmacológicamente activas
Anales de la Real Academia de Ciencias Veterinarias, Vol. 24, Núm. 24, pp. 267-300
2015
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Bond-based bilinear indices for computational discovery of novel trypanosomicidal drug-like compounds through virtual screening
European Journal of Medicinal Chemistry, Vol. 96, pp. 238-244
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Novel solid dispersions of benznidazole: Preparation, dissolution profile and biological evaluation as alternative antichagasic drug delivery system
Experimental Parasitology, Vol. 149, pp. 84-91
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Sequestration of host-CD59 as potential immune evasion strategy of Trichomonas vaginalis
Acta Tropica, Vol. 149, pp. 1-7
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Synthesis and in vitro and in vivo biological evaluation of substituted nitroquinoxalin-2-ones and 2,3-diones as novel trichomonacidal agents
European Journal of Medicinal Chemistry, Vol. 94, pp. 276-283
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The efficacy of 2-nitrovinylfuran derivatives against Leishmania in vitro and in vivo
Memorias do Instituto Oswaldo Cruz, Vol. 110, Núm. 2, pp. 166-173