JOSÉ JAVIER
FERNÁNDEZ RUIZ
Catedrático de universidad
Nadine
Jagerovic
Publicaciones en las que colabora con Nadine Jagerovic (17)
2023
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Thienopyrimidine Derivatives as GPR55 Receptor Antagonists: Insight into Structure-Activity Relationship
ACS Medicinal Chemistry Letters, Vol. 14, Núm. 1, pp. 18-25
2021
2020
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Discovery of Homobivalent Bitopic Ligands of the Cannabinoid CB2 Receptor**
Chemistry - A European Journal, Vol. 26, Núm. 68, pp. 15839-15842
2017
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Corrigendum to “Biological characterization of PM226, a chromenoisoxazole, as a selective CB2 receptor agonist with neuroprotective profile” [Pharmacol. Res. (2016) 110(2016) (205–215)] (S1043661816302080) (10.1016/j.phrs.2016.03.021)
Pharmacological Research
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New pyridazinone-4-carboxamides as new cannabinoid receptor type-2 inverse agonists: Synthesis, pharmacological data and molecular docking
European Journal of Medicinal Chemistry, Vol. 127, pp. 398-412
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Synthesis of a novel CB2 cannabinoid-porphyrin conjugate based on an antitumor chromenopyrazoledione
Journal of Porphyrins and Phthalocyanines, Vol. 21, Núm. 1, pp. 67-76
2016
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Biological characterization of PM226, a chromenoisoxazole, as a selective CB2 receptor agonist with neuroprotective profile
Pharmacological Research, Vol. 110, pp. 205-215
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Chromenopyrazole, a Versatile Cannabinoid Scaffold with in Vivo Activity in a Model of Multiple Sclerosis
Journal of Medicinal Chemistry, Vol. 59, Núm. 14, pp. 6753-6771
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Identification of Novel GPR55 Modulators Using Cell-Impedance-Based Label-Free Technology
Journal of Medicinal Chemistry, Vol. 59, Núm. 5, pp. 1840-1853
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Targeting cannabinoid CB2 receptors in the central nervous system. Medicinal chemistry approaches with focus on neurodegenerative disorders
Frontiers in Neuroscience, Vol. 10, Núm. SEP
2015
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Selective, nontoxic CB2 cannabinoid o-quinone with in vivo activity against triple-negative breast cancer
Journal of Medicinal Chemistry, Vol. 58, Núm. 5, pp. 2256-2264
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Synthesis, pharmacological evaluation and docking studies of pyrrole structure-based CB2 receptor antagonists
European Journal of Medicinal Chemistry, Vol. 101, pp. 651-667
2014
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Combining rimonabant and fentanyl in a single entity: Preparation and pharmacological results
Drug Design, Development and Therapy, Vol. 8, pp. 263-277
2013
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Description of a bivalent cannabinoid ligand with hypophagic properties
Archiv der Pharmazie, Vol. 346, Núm. 3, pp. 171-179
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Novel antiobesity agents: Synthesis and pharmacological evaluation of analogues of Rimonabant and of LH21
Bioorganic and Medicinal Chemistry, Vol. 21, Núm. 7, pp. 1708-1716
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Synthetic cannabinoid quinones: Preparation, in vitro antiproliferative effects and in vivo prostate antitumor activity
European Journal of Medicinal Chemistry, Vol. 70, pp. 111-119
2012
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Chromenopyrazoles: Non-psychoactive and Selective CB 1 Cannabinoid Agonists with Peripheral Antinociceptive Properties
ChemMedChem, Vol. 7, Núm. 3, pp. 452-463