MARÍA ESPERANZA
HERREROS AVILÉS
Profesora asociada
Publicaciones (41) Publicaciones de MARÍA ESPERANZA HERREROS AVILÉS
2021
-
A novel class of fast-acting antimalarial agents: Substituted 15-membered azalides
British Journal of Pharmacology, Vol. 178, Núm. 2, pp. 363-377
-
Barcoded Asaia bacteria enable mosquito in vivo screens and identify novel systemic insecticides and inhibitors of malaria transmission
PLoS Biology, Vol. 19, Núm. 12
-
The antimalarial efficacy and mechanism of resistance of the novel chemotype DDD01034957
Scientific Reports, Vol. 11, Núm. 1
2020
-
Identification of Selective Inhibitors of Plasmodium N-Myristoyltransferase by High-Throughput Screening
Journal of Medicinal Chemistry, Vol. 63, Núm. 2, pp. 591-600
2018
-
A high throughput screen for next-generation leads targeting malaria parasite transmission
Nature Communications, Vol. 9, Núm. 1
-
Erratum for Brunschwig et al., "UCT943, a Next-Generation Plasmodium falciparum PI4K Inhibitor Preclinical Candidate for the Treatment of Malaria" (Antimicrobial Agents and Chemotherapy (2018) 62:9 (e00012-18) DOI: 10.1128/AAC.00012-18)
Antimicrobial Agents and Chemotherapy
-
Gametocytes from K13 propeller mutant plasmodium falciparum clinical isolates demonstrate reduced susceptibility to dihydroartemisinin in the male gamete exflagellation inhibition assay
Antimicrobial Agents and Chemotherapy, Vol. 62, Núm. 12
-
Potent Plasmodium falciparum gametocytocidal compounds identified by exploring the kinase inhibitor chemical space for dual active antimalarials
Journal of Antimicrobial Chemotherapy, Vol. 73, Núm. 5, pp. 1279-1290
-
Synthesis and Structure-Activity Relationships of the Novel Antimalarials 5-Pyridinyl-4(1 H)-Pyridones
Journal of Medicinal Chemistry, Vol. 61, Núm. 8, pp. 3422-3435
-
Uct943, a next-generation plasmodium falciparum pi4k inhibitor preclinical candidate for the treatment of malaria
Antimicrobial Agents and Chemotherapy, Vol. 62, Núm. 9
2017
-
A tetraoxane-based antimalarial drug candidate that overcomes PfK13-C580Y dependent artemisinin resistance
Nature Communications, Vol. 8
-
Hundreds of dual-stage antimalarial molecules discovered by a functional gametocyte screen
Nature Communications, Vol. 8
2016
-
A novel validated assay to support the discovery of new anti-malarial gametocytocidal agents
Malaria Journal, Vol. 15, Núm. 1
-
Transmission-blocking potential of MEFAS, a hybrid compound derived from artesunate and mefloquine
Antimicrobial Agents and Chemotherapy, Vol. 60, Núm. 5, pp. 3145-3147
2015
-
A new Set of chemical starting points with Plasmodium falciparum transmission-blocking potential for antimalarial drug discovery
PLoS ONE, Vol. 10, Núm. 8
-
Imaging-based high-throughput screening assay to identify new molecules with transmission-blocking potential against Plasmodium falciparum female gamete formation
Antimicrobial Agents and Chemotherapy, Vol. 59, Núm. 6, pp. 3298-3305
2013
-
Erratum: Potent antimalarial 4-pyridones with improved physico-chemical properties (Bioorganic and Medicinal Chemistry Letters (2011) 21 (5214-5218))
Bioorganic and Medicinal Chemistry Letters
-
Male and female Plasmodium falciparum mature gametocytes show different responses to antimalarial drugs
Antimicrobial Agents and Chemotherapy, Vol. 57, Núm. 7, pp. 3268-3274
-
Quinolone-3-diarylethers: A new class of antimalarial drug
Science Translational Medicine, Vol. 5, Núm. 177
-
Red blood cells derived from peripheral blood and bone marrow CD34+ human haematopoietic stem cells are permissive to Plasmodium parasites infection
Memorias do Instituto Oswaldo Cruz, Vol. 108, Núm. 6, pp. 801-803